Blar i Bergen Open Research Archive på forfatter "Rekand, Illimar Hugo"
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DrugPred_RNA—A Tool for Structure-Based Druggability Predictions for RNA Binding Sites
Rekand, Illimar Hugo; Brenk, Ruth (Journal article; Peer reviewed, 2021)RNA is an emerging target for drug discovery. However, like for proteins, not all RNA binding sites are equally suited to be addressed with conventional drug-like ligands. To this end, we have developed the structure-based ... -
Structure-based Druggability Predictions of RNA Binding Sites and Design of RNA Ligands
Rekand, Illimar Hugo (Doctoral thesis, 2022-09-15)Den post-antibotiske æraen truer og for å møte denne krisen trengs det tilgang til nye klasser av antibiotika. Ribvoswitcher er cis-genregulerende foldete strukturer av ikke-kodende RNA, som handler gjennom konformasjonsendringer ...